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Synthesis and Antifungal Activities of 2-(N-Arylsulfonylindol-3-yl)-3-aryl-1,3-thiazinan-4-ones

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Synthesis and Antifungal Activities of

2-( N -Arylsulfonylindol-3-yl)-3-aryl-1,3-thiazinan-4-ones

Huan Qu, Rui Zhang, Ying Hu, Yazhen Ke, Zhinan Gao, and Hui Xu*

Laboratory of Pharmaceutical Design & Synthesis, College of Sciences,

Northwest A & F University, Yangling 712100, P. R. China. Fax: +86-29-87091952.

E-mail: orgxuhui@nwsuaf.edu.cn

* Author for correspondence and reprint requests

Z. Naturforsch. 68 c, 77 − 81 (2013); received March 14/June 28, 2012

A series of 2-(N-arylsulfonylindol-3-yl)-3-aryl-1,3-thiazinan-4-one derivatives were syn- thesized and evaluated in vitro against seven phytopathogenic fungi, namely Fusarium graminearum, Alternaria solani, Fusarium oxysporium f. sp. vasinfectum, Alternaria brassi- cae, Valsa mali, Alternaria alternata, and Pyricularia oryzae. Among all derivatives, especially compound 4j exhibited a potential antifungal activity against four phytopathogenic fungi.

Key words: 2-(N-Arylsulfonylindol-3-yl)-3-aryl-1,3-thiazinan-4-ones, Antifungal Activity, Phytopathogenic Fungi

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